SCHEMBL28808185

SCHEMBL28808185

CONC(=O)c1ccc(C2=NOC(c3cc(Cl)cc(Cl)c3)(C(F)(F)F)C2)cn1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 13/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
KDR P35968 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
MAPT P10636 1/20 0.32
BACE2 Q9Y5Z0 2/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29724107 1.00 BACE1 (0.34) BACE1CA1CA2KDRTDP1
SCHEMBL12449485 0.86 MAP4K4 (0.38) BACE1CA1CA2KDM4E
SCHEMBL28947412 0.85 BACE1 (0.33) BACE1CA1CA2BACE2APP
SCHEMBL29724089 0.85 BACE1 (0.33) BACE1CA1CA2BACE2APP
SCHEMBL28808904 0.82 CA1 (0.35) CA1CA2
SCHEMBL28808902 0.81 HIF1A (0.35)
SCHEMBL740580 0.80 KDM4E (0.48) CA1CA2MAPTKDM4E
SCHEMBL29700184 0.80 KCNH2 (0.38) BACE1
SCHEMBL1611226 0.79 NPC1 (0.33) MAPTKDM4E
SCHEMBL3358580 0.78 RECQL (0.32) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114853748-A Trifluoromethyl-containing isoxazoline derivative, and preparation method and application thereof 武汉工程大学 2022-08-05 CN disclosed