SCHEMBL28808283

SCHEMBL28808283

CC(C)(C)OC(=O)c1cc2ccc(N)cc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.51
ALOX15 P16050 3/20 0.45
KDM4E B2RXH2 3/20 0.41
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
EIF4A3 P38919 1/20 0.39
FLT3 P36888 3/20 0.39
RET P07949 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3494717 0.88 HRH4 (0.51) HRH4KDM4ELMNATP53L3MBTL1
SCHEMBL654862 0.83 HRH4 (0.55) HRH4ALOX15KDM4ELMNATP53
SCHEMBL17092514 0.83 HRH4 (0.55) HRH4ALOX15KDM4ELMNATP53
SCHEMBL20612119 0.82 HRH4 (0.51) HRH4ALOX15KDM4ELMNATP53
Hydrochloric Acid SCHEMBL23045607 0.82 HRH4 (0.53) HRH4ALOX15KDM4ELMNATP53
Hydrochloric Acid SCHEMBL31383573 0.82 HRH4 (0.53) HRH4ALOX15KDM4ELMNATP53
SCHEMBL6947975 0.81 HRH3 (0.52) ALOX15KDM4ELMNATP53L3MBTL1
SCHEMBL29496122 0.80 KDM4E (0.63) KDM4ELMNATP53L3MBTL1ALDH1A1
SCHEMBL318243 0.80 KDM4E (0.63) KDM4ELMNATP53L3MBTL1ALDH1A1
SCHEMBL20612118 0.80 RAB9A (0.48) ALOX15KDM4ELMNAL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728914-B Dioxopiperazine derivative, preparation method thereof and application thereof in medicines 深圳信立泰药业股份有限公司 2023-05-12 CN disclosed
CN-114728914-A Dioxopiperazine derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2022-07-08 CN disclosed