SCHEMBL28810458

SCHEMBL28810458

NC(=O)OC1CCN(C(=O)C2(c3ccccc3)CCN(c3cc(Cl)nnc3N)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 3/20 0.43
KCNH2 Q12809 2/20 0.43
HSD11B1 P28845 10/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR1 P21554 3/20 0.36
GPR55 Q9Y2T6 3/20 0.36
CNR2 P34972 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23302103 0.86 PBRM1 (0.52)
SCHEMBL23301263 0.84 KCNH2 (0.43) OPRD1KCNH2HSD11B1MEN1KMT2A
SCHEMBL29943255 0.83 OPRD1 (0.51) OPRD1KCNH2MEN1KMT2ASMN1; SMN2
SCHEMBL23301640 0.83 OPRD1 (0.51) OPRD1KCNH2MEN1KMT2ASMN1; SMN2
SCHEMBL29943128 0.82 CKS1B (0.42) OPRD1KCNH2HSD11B1KMT2ACNR1
SCHEMBL23037203 0.81 PBRM1 (0.38) MEN1KMT2ASMN1; SMN2ALDH1A1LMNA
SCHEMBL28810427 0.81 SMARCA2 (0.54) OPRD1KCNH2HSD11B1TSHR
SCHEMBL29943226 0.81 SMARCA2 (0.54) OPRD1KCNH2HSD11B1TSHR
SCHEMBL23301272 0.77 SMARCA2 (0.47) OPRD1KCNH2HSD11B1TSHR
SCHEMBL29942944 0.77 SMARCA2 (0.47) OPRD1KCNH2HSD11B1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728936-A Bifunctional compounds for the treatment of cancer 豪夫迈·罗氏有限公司 2022-07-08 CN disclosed