SCHEMBL28810567

SCHEMBL28810567

Clc1ccc2cc(Br)nc(Cl)c2c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
NR4A2 P43354 2/20 0.34
NOS1 P29475 1/20 0.34
DYRK1A Q13627 1/20 0.34
LMNA P02545 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CHEK1 O14757 1/20 0.33
S1PR4 O95977 1/20 0.33
KMT2A Q03164 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
TYMS P04818 3/20 0.33
POLB P06746 1/20 0.32
CMA1 P23946 1/20 0.32
AHR P35869 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PIM1 P11309 1/20 0.32
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11792799 0.78 CYP2A6 (0.39) CYP2A6NR4A2NOS1DYRK1ALMNA
SCHEMBL374938 0.77 ALDH1A1 (0.39) CYP2A6LMNAALDH1A1L3MBTL1
SCHEMBL3964092 0.76 CCR1 (0.38) CYP2A6NR4A2NOS1DYRK1ALMNA
SCHEMBL4387539 0.75 POLB (0.48) CYP2A6NR4A2ALDH1A1TYMSPOLB
SCHEMBL30800385 0.71 HTT (0.38) CYP2A6NR4A2NOS1ALDH1A1KMT2A
SCHEMBL28962504 0.71 HTT (0.38) CYP2A6NR4A2NOS1ALDH1A1KMT2A
SCHEMBL28327302 0.71 S1PR4 (0.40) CYP2A6NR4A2NOS1S1PR4TYMS
SCHEMBL16008294 0.71 CYP2A6 (0.39) CYP2A6DYRK1ALMNAALDH1A1CHEK1
SCHEMBL28656122 0.69 ALDH1A1 (0.41) NR4A2LMNAALDH1A1KDM4EHTT
SCHEMBL28130492 0.69 NT5E (0.46) NR4A2LMNAALDH1A1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103562199-A Tripeptides incorporating deuterium as inhibitors of hepatitis c virus BRISTOL MYERS SQUIBB CO 2014-02-05 CN disclosed