SCHEMBL28811700

SCHEMBL28811700

CC(C)(C)OC(=O)N1CCC(Nc2ccc3c(c2)CC(=O)N3)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
NPC1 O15118 2/20 0.60
RAB9A P51151 2/20 0.60
MAPT P10636 2/20 0.60
MAPK1 P28482 1/20 0.60
HTT P42858 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
CRBN Q96SW2 3/20 0.58
DDB1 Q16531 2/20 0.54
PTPN2 P17706 1/20 0.49
PTPN1 P18031 1/20 0.49
PTPN6 P29350 1/20 0.49
SMYD3 Q9H7B4 1/20 0.47
GRIN1 Q05586 2/20 0.46
GRIN2B Q13224 2/20 0.46
GRIN2D O15399 1/20 0.46
GRIN3B O60391 1/20 0.46
GRIN2A Q12879 1/20 0.46
GRIN2C Q14957 1/20 0.46
GRIN3A Q8TCU5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3290755 0.86 KDM4E (0.55) ALDH1A1MAPTHTTSMYD3GRIN1
SCHEMBL17591942 0.84 SMYD3 (0.62) CRBNSMYD3
SCHEMBL6832459 0.82 SYK (0.57) ALDH1A1NPC1RAB9AMAPTMAPK1
SCHEMBL12431387 0.82 SMYD3 (0.59) ALDH1A1HTTCRBNSMYD3
SCHEMBL16047746 0.82 CRBN (0.58) MAPTHTTCRBNDDB1PTPN2
SCHEMBL30847573 0.82 CRBN (0.58) MAPTHTTCRBNDDB1PTPN2
SCHEMBL13586867 0.81 POLB (0.52) MAPTSMYD3GRIN1GRIN2BGRIN2D
SCHEMBL10269535 0.81 ALDH1A1 (0.63) ALDH1A1NPC1RAB9AMAPTMAPK1
SCHEMBL12853755 0.78 ALDH1A1 (0.63) ALDH1A1NPC1RAB9AMAPTMAPK1
SCHEMBL4115820 0.78 ALDH1A1 (0.77) ALDH1A1NPC1RAB9AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107072205-B SMYD inhibitors EPIZYME股份有限公司 2022-07-15 CN disclosed