SCHEMBL28811771

SCHEMBL28811771

CN1CCc2c(Br)cc(I)cc2C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.40
MAOB P27338 4/20 0.40
SLC6A4 P31645 1/20 0.39
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
DRD1 P21728 2/20 0.33
DRD5 P21918 2/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29843380 1.00 MAOA (0.40) MAOAMAOBSLC6A4ADRA2AADRA2B
SCHEMBL25840894 0.79 MAOA (0.40) MAOAMAOBSLC6A4ADRA2AADRA2B
SCHEMBL8185029 0.79 MAOA (0.40) MAOAMAOBSLC6A4KDM4EMAPT
SCHEMBL24040089 0.79 MAOA (0.40) MAOAMAOBSLC6A4ADRA2AADRA2B
SCHEMBL29557955 0.79 MAOA (0.40) MAOAMAOBSLC6A4ADRA2AADRA2B
SCHEMBL8176774 0.73 GRIA1 (0.49) MAOAMAOBMAPTALDH1A1
SCHEMBL16076617 0.71 MAOA (0.57) MAOAMAOBADRA2AADRA2BADRA2C
SCHEMBL22450600 0.71 MAOA (0.55) MAOAMAOBSLC6A4ADRA2AADRA2B
SCHEMBL29507157 0.70 MAOA (0.41) MAOAMAOBSLC6A4ADRA2AADRA2B
SCHEMBL22858691 0.70 MAOA (0.41) MAOAMAOBSLC6A4ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114853730-B Compounds used as HPK1 kinase inhibitor, preparation method and application thereof 中国药科大学 2024-03-26 CN disclosed
CN-114853730-A Compound used as HPK1 kinase inhibitor and preparation method and application thereof 中国药科大学 2022-08-05 CN disclosed