SCHEMBL28813643

SCHEMBL28813643

CC(=O)Nn1ccc(C#N)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.38
IDO1 P14902 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SETDB1 Q15047 1/20 0.36
ALDH1A1 P00352 2/20 0.33
DYRK1A Q13627 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
EGLN2 Q96KS0 1/20 0.33
MAPT P10636 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
AR P10275 1/20 0.32
PGR P06401 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651804 0.72 NOTUM (0.36) SETDB1ALDH1A1MAPTCA1CA2
SCHEMBL28980345 0.65 DYRK1A (0.40) KDM1ASETDB1ALDH1A1DYRK1AKDM4E
Ciapilome SCHEMBL2110362 0.65 ELANE (0.35) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL28582333 0.64 PARP15 (0.37) CA1CA2PGR
SCHEMBL1780017 0.63
SCHEMBL7041642 0.63
SCHEMBL5610745 0.62
SCHEMBL27367482 0.62 TSHR (0.39) ALDH1A1KDM4ECA2LOXL2
SCHEMBL24621213 0.62 AKR1B1 (0.50) L3MBTL1ALDH1A1KDM4EMAPTAR
SCHEMBL31241488 0.62 POLB (0.55) L3MBTL1ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103864661-A Synthesis process of 2-amino-3-cyano pyrrole derivatives Hunan huateng pharmaceutical co ltd 2014-06-18 CN disclosed