SCHEMBL28813848

SCHEMBL28813848

Cn1ncc([N+](=O)[O-])c1N1CCC(N(N)C(=O)O)CC(O)C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.32
JAK3 P52333 2/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
PKM P14618 1/20 0.32
KMT2A Q03164 4/20 0.31
LMNA P02545 1/20 0.31
MEN1 O00255 3/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
MAPT P10636 1/20 0.31
CTPS1 P17812 1/20 0.31
PIM1 P11309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27980042 0.85 ALDH1A1 (0.36) GAAPKMKMT2ALMNAMEN1
SCHEMBL28813927 0.82 CTPS1 (0.33) GAAPKMKMT2AMEN1POLB
SCHEMBL14801332 0.82 PIM1 (0.35) KMT2ALMNAMEN1ALDH1A1MAPT
SCHEMBL2515867 0.81 MEN1 (0.39) GAAPKMKMT2ALMNAMEN1
SCHEMBL2515869 0.81 MEN1 (0.39) GAAPKMKMT2ALMNAMEN1
SCHEMBL2522631 0.81 MEN1 (0.39) GAAPKMKMT2ALMNAMEN1
SCHEMBL27980071 0.81 GAA (0.34) GAAPKMKMT2AMEN1ALDH1A1
SCHEMBL28813851 0.79 GAA (0.35) GAAPKMKMT2AMEN1POLB
SCHEMBL14686310 0.79 KMT2A (0.42) GAAPKMKMT2ALMNAMEN1
SCHEMBL14800963 0.77 MEN1 (0.43) GAAPKMKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103987707-A Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use HOFFMANN LA ROCHE 2014-08-13 CN disclosed