SCHEMBL28814166

SCHEMBL28814166

Nc1ncc(-c2cc(CC3CC3)[nH]n2)c(N)n1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CG P48736 1/20 0.37
PIK3C3 Q8NEB9 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
DHFR P00374 6/20 0.35
FGFR1 P11362 4/20 0.33
SRC P12931 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27983193 0.79 DHFR (0.39) PIK3CAPIK3CDPIK3CGPIK3C3PI4KB
SCHEMBL4457723 0.76 HCAR2 (0.43) PIK3CADHFRADORA2AADORA1
SCHEMBL30065933 0.75 NPC1 (0.50) PIK3CADHFRFGFR1SRC
SCHEMBL3663141 0.75 NPC1 (0.50) PIK3CADHFRFGFR1SRC
SCHEMBL28664537 0.74 MKNK1 (0.40) PIK3CADHFRADORA2AADORA1
SCHEMBL27983086 0.70 MKNK1 (0.34) PIK3CAPIK3CDPIK3CGPIK3C3PI4KB
SCHEMBL28814284 0.69 PIK3CA (0.35) PIK3CADHFRADORA2AADORA1
SCHEMBL27983380 0.69 PIK3CA (0.35) PIK3CADHFRADORA2AADORA1
SCHEMBL27983385 0.69 PIK3CA (0.35) PIK3CADHFRADORA2AADORA1
SCHEMBL28649163 0.69 PIK3CA (0.40) PIK3CADHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104024248-A SERINE/THREONINE PAK1 INHIBITORS HOFFMANN LA ROCHE 2014-09-03 CN disclosed