SCHEMBL28815566

SCHEMBL28815566

NC(=O)c1ccc(-c2cccnc2)c(-c2cccnc2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 8/20 0.51
MKNK2 Q9HBH9 8/20 0.51
ADORA2A P29274 1/20 0.51
ADORA2B P29275 1/20 0.51
IKBKB O14920 1/20 0.47
F7 P08709 1/20 0.46
F3 P13726 1/20 0.46
SARM1 Q6SZW1 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.46
SIRT6 Q8N6T7 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
SIRT5 Q9NXA8 1/20 0.46
SIRT4 Q9Y6E7 1/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
LMNA P02545 1/20 0.46
CYP2C19 P33261 1/20 0.46
SCN9A Q15858 3/20 0.43
PKN1 Q16512 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29504504 1.00 MKNK1 (0.51) MKNK1MKNK2ADORA2AADORA2BIKBKB
SCHEMBL29504529 0.87 CYP2A6 (0.54) MKNK1MKNK2ADORA2AADORA2BIKBKB
Hydrochloric Acid SCHEMBL29504512 0.86 CYP2A6 (0.52) MKNK1MKNK2ADORA2AADORA2BIKBKB
SCHEMBL29911882 0.85 MKNK1 (0.52) MKNK1MKNK2IKBKBF7F3
SCHEMBL28826508 0.84 IKBKB (0.54) MKNK1MKNK2IKBKBF7F3
SCHEMBL5320803 0.83 CYP3A4 (0.55) MKNK1MKNK2IKBKBF7F3
Formic Acid SCHEMBL29911825 0.80 MKNK1 (0.48) MKNK1MKNK2IKBKBF7F3
SCHEMBL7090661 0.80 ALDH1A1 (0.47) MKNK2ADORA2ALMNAALDH1A1
SCHEMBL31188541 0.78 MKNK1 (0.58) MKNK1MKNK2CYP1A2CYP3A4LMNA
SCHEMBL29505512 0.78 SCN9A (0.59) MKNK1MKNK2IKBKBF7F3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104125947-A Heterocyclic urea compounds BIOTA EUROPE LTD 2014-10-29 CN disclosed