SCHEMBL28817261

SCHEMBL28817261

N#Cc1ccc2c(ccn2-c2nc(Cl)ncc2C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 7/20 0.46
ENPP3 O14638 1/20 0.38
GRM2 Q14416 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
RPS6KA5 O75582 6/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
CDK2 P24941 3/20 0.36
MAP3K14 Q99558 1/20 0.36
TRPV4 Q9HBA0 1/20 0.35
RPS6KA4 O75676 1/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30007251 1.00 CDC7 (0.46) CDC7ENPP3GRM2FFAR4RPS6KA5
SCHEMBL30750938 0.91 CDC7 (0.46) CDC7GRM2RPS6KA5CDK2MAP3K14
SCHEMBL28617905 0.79 RPS6KA5 (0.47) CDC7RPS6KA5CDK2RPS6KA4
SCHEMBL29651176 0.79 RPS6KA5 (0.47) CDC7RPS6KA5CDK2RPS6KA4
SCHEMBL27253692 0.77 RPS6KA5 (0.41) RPS6KA5RPS6KA4
SCHEMBL17682937 0.76 GRM2 (0.36) GRM2TRPV4PSEN1PSEN2APH1B
SCHEMBL19540762 0.73 RARG (0.37) GRM2TRPV4PSEN1PSEN2APH1B
SCHEMBL19254673 0.73 GRM2 (0.36) GRM2CDK2TRPV4PSEN1PSEN2
SCHEMBL30394203 0.73 ENPP3 (0.48) CDC7ENPP3GRM2FFAR4CDK2
SCHEMBL27400872 0.73 ENPP3 (0.48) CDC7ENPP3GRM2FFAR4CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907407-A Inhibitors of cyclin dependent kinase 7(CDK7) 江苏先声药业有限公司 2022-08-16 CN disclosed