SCHEMBL28818554

SCHEMBL28818554

CC(C)C(C)(C(=O)O)c1ccc(C(C)(C(=O)O)C(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.50
CYP2C9 P11712 2/20 0.50
HIF1A Q16665 2/20 0.50
CYP1A2 P05177 4/20 0.45
CYP2C19 P33261 1/20 0.39
SRD5A2 P31213 1/20 0.38
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
NR1H4 Q96RI1 2/20 0.36
MAPT P10636 1/20 0.35
HDAC1 Q13547 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ESR1 P03372 1/20 0.34
CYP3A4 P08684 1/20 0.34
ESR2 Q92731 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20425516 0.94 SRD5A2 (0.47) CYP2D6CYP2C9HIF1ACYP1A2SRD5A2
SCHEMBL3495875 0.92 CYP2D6 (0.44) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19
SCHEMBL3304253 0.91 CYP1A2 (0.57) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19
SCHEMBL9966556 0.90 CYP2D6 (0.43) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19
SCHEMBL11168281 0.90 KMT2A (0.50) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19
SCHEMBL28727642 0.89 CYP1A2 (0.55) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19
SCHEMBL28727574 0.89 CYP1A2 (0.55) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19
SCHEMBL5317094 0.88 MAPT (0.49) MAPTALDH1A1
SCHEMBL30091181 0.85 PTGS1 (0.50) CYP2C9ESR1RARB
SCHEMBL8984193 0.85 CES2 (0.41) CYP2D6CYP2C9HIF1ACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901653-A Novel amide derivatives useful as diacylglycerol acyltransferase 2 inhibitors and uses thereof 株式会社LG化学 2022-08-12 CN disclosed