SCHEMBL28819986

SCHEMBL28819986

O=c1[nH]nc(CCBr)cc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 7/20 0.44
IDO1 P14902 1/20 0.36
AR P10275 1/20 0.35
NOTUM Q6P988 2/20 0.33
PRMT5 O14744 2/20 0.32
WDR77 Q9BQA1 2/20 0.32
AKR1B1 P15121 1/20 0.31
ALDH1A1 P00352 2/20 0.31
GAA P10253 2/20 0.31
DAO P14920 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
HPGD P15428 1/20 0.31
ENPP1 P22413 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15633341 0.86 TIPARP (0.40) TIPARPIDO1ARNOTUMPRMT5
SCHEMBL30859999 0.83 TIPARP (0.44) TIPARPIDO1ARNOTUMALDH1A1
SCHEMBL30859849 0.79 TIPARP (0.40) TIPARPIDO1ARNOTUMPRMT5
SCHEMBL24968908 0.75 TIPARP (0.43) TIPARPIDO1AR
SCHEMBL30851298 0.74 TIPARP (0.42) TIPARPIDO1ARNOTUMPRMT5
SCHEMBL30507321 0.74 TIPARP (0.43) TIPARPIDO1NOTUMPRMT5WDR77
SCHEMBL31464989 0.73 NOTUM (0.40) TIPARPIDO1ARNOTUMPRMT5
SCHEMBL24739044 0.69 NOTUM (0.40) ARNOTUMALDH1A1GAA
SCHEMBL15633366 0.69 NOTUM (0.43) TIPARPARNOTUMPRMT5WDR77
SCHEMBL24739443 0.69 BACE1 (0.37) TIPARPARNOTUMPRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104822670-A 5-phenoxy-3h-pyrimidin-4-one derivatives and their use as HIV reverse transcriptase inhibitors MERCK SHARP & DOHME 2015-08-05 CN disclosed