Indazole

Indazole

SCHEMBL28820118

Nc1cccc(-c2ccccc2)c1.c1ccc2[nH]ncc2c1

nearest known ligand 0.61

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 1/20 0.61
DYRK3 O43781 1/20 0.61
CLK1 P49759 1/20 0.61
CLK2 P49760 1/20 0.61
CLK3 P49761 1/20 0.61
GSK3B P49841 1/20 0.61
CDK5 Q00535 1/20 0.61
DYRK1A Q13627 1/20 0.61
CDK5R1 Q15078 1/20 0.61
DYRK2 Q92630 1/20 0.61
CLK4 Q9HAZ1 1/20 0.61
DYRK1B Q9Y463 1/20 0.61
HSP90AA1 P07900 1/20 0.59
IDO1 P14902 1/20 0.59
CDK2 P24941 1/20 0.59
MAOA P21397 1/20 0.56
KDM4E B2RXH2 4/20 0.53
MEN1 O00255 3/20 0.53
MAPT P10636 3/20 0.53
KMT2A Q03164 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8266373 0.84 FGFR1 (0.70) FGFR1DYRK3CLK1CLK2CLK3
Indazole SCHEMBL7371212 0.79 HSP90AA1 (0.95) FGFR1DYRK3CLK1CLK2CLK3
Indazole SCHEMBL27944553 0.78 HSP90AA1 (0.54) FGFR1DYRK3CLK1CLK2CLK3
Indazole SCHEMBL27558509 0.77 HSP90AA1 (0.91) FGFR1DYRK3CLK1CLK2CLK3
Indazole SCHEMBL1221882 0.77 HSP90AA1 (1.00) FGFR1DYRK3CLK1CLK2CLK3
Indazole SCHEMBL6295 0.77
Indazole SCHEMBL29355507 0.77
SCHEMBL2455100 0.76 GSK3B (1.00) FGFR1DYRK3CLK1CLK2CLK3
SCHEMBL2460902 0.76 FGFR1 (1.00) FGFR1DYRK3CLK1CLK2CLK3
Anthracene SCHEMBL15271626 0.75 HSP90AA1 (0.86) FGFR1DYRK3CLK1CLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104725319-A 1H-indazole-3-aminobphenyl urea compound with anti-tumor activity as well as preparation method and application of 1H-indazole-3-aminobphenyl urea compound UNIV XI AN JIAOTONG 2015-06-24 CN disclosed