SCHEMBL28820802

SCHEMBL28820802

COc1cc2ccc(Nc3ccc(F)c(Cl)c3)nc2cc1OC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.50
CSF1R P07333 1/20 0.49
ERBB2 P04626 8/20 0.48
KDR P35968 3/20 0.48
AURKA O14965 1/20 0.48
INSR P06213 1/20 0.48
FBP1 P09467 1/20 0.48
PDGFRB P09619 1/20 0.48
FLT4 P35916 1/20 0.48
CLK1 P49759 1/20 0.48
EPHB4 P54760 1/20 0.48
TEK Q02763 1/20 0.48
AURKB Q96GD4 1/20 0.48
MAPT P10636 2/20 0.46
POLB P06746 1/20 0.46
HDAC3 O15379 3/20 0.44
HDAC4 P56524 3/20 0.44
HDAC1 Q13547 3/20 0.44
HDAC7 Q8WUI4 3/20 0.44
HDAC2 Q92769 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29881841 1.00 EGFR (0.50) EGFRCSF1RERBB2KDRAURKA
SCHEMBL27896795 0.85 EGFR (0.51) EGFRCSF1RERBB2KDRAURKA
SCHEMBL30968993 0.84 EGFR (0.53) EGFRCSF1RERBB2KDRAURKA
SCHEMBL28820741 0.84 RAF1 (0.50) EGFRCSF1RERBB2KDRAURKA
SCHEMBL29881898 0.84 RAF1 (0.50) EGFRCSF1RERBB2KDRAURKA
SCHEMBL28820762 0.82 SLC2A1 (0.44) EGFRKDRPDGFRBMAPTPOLB
SCHEMBL28820840 0.81 EGFR (0.55) EGFRERBB2KDRAURKAINSR
SCHEMBL29881732 0.81 EGFR (0.55) EGFRERBB2KDRAURKAINSR
SCHEMBL29882028 0.78 EGFR (0.67) EGFRCSF1RKDR
SCHEMBL30968994 0.78 EGFR (0.82) EGFRERBB2KDRAURKAINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114907261-B 2-phenylaminoquinoline derivative, preparation method and application thereof 湖南中医药大学 2023-10-27 CN disclosed
CN-114907261-A 2-phenylamino quinoline derivative and preparation method and application thereof 湖南中医药大学 2022-08-16 CN disclosed