SCHEMBL28822758

SCHEMBL28822758

O=C(O)Cc1cccc2c(=O)cc(-c3cccnc3C(F)(F)F)oc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.40
CYP1A1 P04798 7/20 0.40
CYP1B1 Q16678 7/20 0.40
CYP2D6 P10635 3/20 0.40
DHODH Q02127 1/20 0.39
GLA P06280 1/20 0.39
STING1 Q86WV6 1/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2C19 P33261 3/20 0.39
STAT6 P42226 1/20 0.39
KDM4E B2RXH2 3/20 0.37
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
TSHR P16473 1/20 0.36
PRKDC P78527 1/20 0.36
CD38 P28907 1/20 0.36
PPARG P37231 1/20 0.35
NR1H2 P55055 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2149236 0.84 CYSLTR1 (0.49) CYP1A2CYP1A1CYP1B1CYP2D6DHODH
SCHEMBL2529900 0.80 CYP1A1 (0.43) CYP1A2CYP1A1CYP1B1CYP2D6DHODH
SCHEMBL9330744 0.79 CYP1A2 (0.58) CYP1A2CYP1A1CYP1B1CYP2D6GLA
SCHEMBL28822757 0.78 CYP3A4 (0.48) CYP1A2CYP1A1CYP1B1CYP2D6DHODH
SCHEMBL2148915 0.78 KDM4E (0.43) CYP1A2CYP1A1CYP1B1DHODHCYP3A4
SCHEMBL9329003 0.78 CYP1A2 (0.48) CYP1A2CYP1A1CYP1B1CYP2D6GLA
SCHEMBL7082926 0.78 CYP1A2 (0.59) CYP1A2CYP1A1CYP1B1CYP2D6GLA
SCHEMBL12835307 0.78 CYP3A4 (0.60) CYP1A2CYP1A1CYP1B1CYP2D6GLA
SCHEMBL7086520 0.77 CYP1A2 (0.55) CYP1A2CYP1A1CYP1B1CYP2D6GLA
SCHEMBL7085772 0.77 CYP3A4 (0.48) CYP1A2CYP1A1CYP1B1CYP2D6GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105198872-A Chromenone analogs as sirtuin modulators SIRTRIS PHARMACEUTICALS INC 2015-12-30 CN disclosed
CN-102227417-B Chromenone analogs as sirtuin modulators SIRTRIS PHARMACEUTICALS, INC. (US) 2015-09-16 CN disclosed