SCHEMBL28822945

SCHEMBL28822945

N#Cc1nc(-c2ccc(Cl)cc2)c(-c2ccccc2)nc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.53
LMNA P02545 3/20 0.53
GAA P10253 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
ADORA1 P30542 10/20 0.52
ADORA2A P29274 9/20 0.52
USP8 P40818 1/20 0.50
ADORA2B P29275 1/20 0.50
DPP4 P27487 1/20 0.48
ERBB2 P04626 1/20 0.47
HPGD P15428 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.45
GRM5 P41594 2/20 0.45
ALDH1A1 P00352 3/20 0.44
HTT P42858 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
THRB P10828 1/20 0.44
GLA P06280 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28822972 1.00 KDM4E (0.53) KDM4ELMNAGAAL3MBTL1ADORA1
SCHEMBL28823015 0.90 USP8 (0.58) KDM4ELMNAADORA1ADORA2AUSP8
SCHEMBL28949045 0.88 ADORA1 (0.66) ADORA1ADORA2AUSP8ADORA2BDPP4
SCHEMBL28823023 0.88 ADORA1 (0.66) ADORA1ADORA2AUSP8ADORA2BDPP4
SCHEMBL28822974 0.84 ADORA1 (0.61) KDM4ELMNAADORA1ADORA2AUSP8
SCHEMBL28823036 0.84 ADORA1 (0.61) KDM4EGAAADORA1ADORA2AUSP8
SCHEMBL28822973 0.84 USP8 (0.57) KDM4ELMNAL3MBTL1ADORA1ADORA2A
SCHEMBL28822976 0.84 USP8 (0.57) KDM4ELMNAL3MBTL1ADORA1ADORA2A
SCHEMBL20666626 0.83 ADORA2A (0.62) KDM4ELMNAL3MBTL1ADORA1ADORA2A
SCHEMBL4678518 0.81 ERBB2 (0.61) KDM4ELMNAGAAL3MBTL1USP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114644597-B Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2023-11-21 CN claimed
CN-114644597-A Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2022-06-21 CN claimed
CN-114644597-B Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2023-11-21 CN disclosed
CN-114644597-A Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2022-06-21 CN disclosed