SCHEMBL28949045

SCHEMBL28949045

N#Cc1nc(-c2cccc(Cl)c2)c(-c2ccccc2)nc1N

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 13/20 0.66
ADORA2A P29274 13/20 0.66
ADORA2B P29275 6/20 0.66
DPP4 P27487 1/20 0.50
USP8 P40818 1/20 0.48
GRM5 P41594 2/20 0.47
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28823023 1.00 ADORA1 (0.66) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL28822972 0.88 KDM4E (0.53) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL28822945 0.88 KDM4E (0.53) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL28823015 0.87 USP8 (0.58) ADORA1ADORA2AADORA2BUSP8
SCHEMBL28822957 0.82 ADORA1 (0.56) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL28822967 0.82 ADORA1 (0.56) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL28822976 0.81 USP8 (0.57) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL28822973 0.81 USP8 (0.57) ADORA1ADORA2AADORA2BDPP4USP8
SCHEMBL20667474 0.81 ADORA2A (0.58) ADORA1ADORA2AADORA2B
SCHEMBL20666626 0.81 ADORA2A (0.62) ADORA1ADORA2AADORA2BUSP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114644597-B Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2023-11-21 CN claimed
CN-114644597-A Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2022-06-21 CN claimed
CN-114644597-B Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2023-11-21 CN disclosed
CN-114644597-A Tetra-substituted pyrazine derivative and preparation method and application thereof 南京农业大学 2022-06-21 CN disclosed