SCHEMBL28824034

SCHEMBL28824034

O=C(O)c1cnnn1-c1ccc(-c2ccccc2)c(-c2cncs2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAUR Q03405 1/20 0.37
KDR P35968 1/20 0.36
HSP90AA1 P07900 2/20 0.35
NPC1 O15118 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHEK2 O96017 2/20 0.35
CHEK1 O14757 1/20 0.35
PIK3CD O00329 1/20 0.34
TSHR P16473 1/20 0.34
F2 P00734 2/20 0.34
F10 P00742 2/20 0.34
PRSS1 P07477 2/20 0.34
PRSS2 P07478 2/20 0.34
PRSS3 P35030 2/20 0.34
MAPK9 P45984 2/20 0.33
PIM1 P11309 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824031 0.91 PLAUR (0.38) PLAURKDRHSP90AA1NPC1NFKB1
SCHEMBL28824104 0.83 MAPK10 (0.47) HSP90AA1NPC1NFKB1RAB9ANFKB2
SCHEMBL28949291 0.82 KMO (0.42) MAPK9MAPK10CA9PTGS2ALDH1A1
SCHEMBL28824080 0.81 NPC1 (0.40) HSP90AA1NPC1NFKB1RAB9ANFKB2
SCHEMBL28824139 0.80 PTGDR2 (0.42) KDRHSP90AA1NPC1NFKB1RAB9A
SCHEMBL28823986 0.79 FOLH1 (0.44) HSP90AA1NPC1NFKB1RAB9ANFKB2
SCHEMBL28949290 0.78 DHODH (0.46) HSP90AA1NPC1NFKB1RAB9ANFKB2
SCHEMBL28824033 0.78 PTGS1 (0.42) HSP90AA1NPC1NFKB1RAB9ANFKB2
SCHEMBL28824039 0.78 CA1 (0.44) HSP90AA1NPC1NFKB1RAB9ANFKB2
SCHEMBL28824007 0.78 NPC1 (0.39) HSP90AA1NPC1NFKB1RAB9ANFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929676-A Heterocyclic carboxylate compounds as glycolate oxidase inhibitors 紫丁香疗法有限公司 2022-08-19 CN disclosed