SCHEMBL28824366

SCHEMBL28824366

CC(C)(C)OC(=O)N1Cc2ccsc2C1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.48
NR1H2 P55055 3/20 0.47
MAPK1 P28482 1/20 0.47
HDAC1 Q13547 1/20 0.45
NAMPT P43490 3/20 0.43
DDB1 Q16531 2/20 0.42
CRBN Q96SW2 2/20 0.42
GPR119 Q8TDV5 3/20 0.42
ADORA1 P30542 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
USP2 O75604 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL976218 0.87 ESR2 (0.58) ESR2NR1H2MAPK1NAMPTADORA1
SCHEMBL1015935 0.87 ESR2 (0.58) ESR2NR1H2MAPK1NAMPTGPR119
SCHEMBL7795095 0.84 ESR2 (0.49) ESR2NR1H2MAPK1ADORA1KDM4E
SCHEMBL3005376 0.79 ESR2 (0.52) ESR2NR1H2MAPK1GPR119ADORA1
SCHEMBL29676965 0.78 MAPK1 (0.64) ESR2NR1H2MAPK1HDAC1NAMPT
SCHEMBL5183098 0.78 MAPK1 (0.64) ESR2NR1H2MAPK1HDAC1NAMPT
SCHEMBL9182719 0.77 ESR2 (0.49) ESR2NR1H2MAPK1HDAC1NAMPT
SCHEMBL30309375 0.76 PDE4B (0.40) ESR2NR1H2MAPK1NAMPTGPR119
SCHEMBL21807285 0.75 MAPK1 (0.52) ESR2NR1H2MAPK1HDAC1NAMPT
SCHEMBL30816257 0.75 HDAC1 (0.45) ESR2NR1H2MAPK1HDAC1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105461733-A (2,4-dihydroxy-5-isopropylphenyl)(4,6-dihydro-5H-thieno[2,3-c]pyrrol-5-yl)ketone derivative, preparation and uses thereof SHANGHAI HANSEN BIOLOGICAL MEDICINE SCIENCE & TECH CO LTD 2016-04-06 CN disclosed