SCHEMBL28824587

SCHEMBL28824587

Nc1cc(-c2nccs2)cs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.47
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
NOS1 P29475 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP2A6 P11509 1/20 0.43
SMPD3 Q9NY59 1/20 0.42
HSP90AA1 P07900 1/20 0.42
ADRB2 P07550 1/20 0.40
CHEK2 O96017 1/20 0.39
ADORA2A P29274 3/20 0.39
HDAC2 Q92769 2/20 0.38
ADORA1 P30542 2/20 0.38
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2552971 0.72 PDPK1 (0.44) PDPK1LOXL2CYP2A6SMPD3HSP90AA1
SCHEMBL3885226 0.71 LOXL2 (0.66) PDPK1LOXL2ALDH1A1TSHRNOS1
SCHEMBL722198 0.71 PDPK1 (0.77) PDPK1LOXL2ALDH1A1TSHRNOS1
SCHEMBL1068648 0.71 LOXL2 (0.55) PDPK1LOXL2ALDH1A1TSHRNOS1
SCHEMBL1653986 0.70 PDPK1 (0.68) PDPK1LOXL2ALDH1A1HSD17B10CYP2A6
SCHEMBL102331 0.69 PDPK1 (0.59) PDPK1LOXL2ALDH1A1TSHRNOS1
Hydrochloric Acid SCHEMBL15911351 0.69 PIK3CD (0.39) ALDH1A1TSHRNOS1HSD17B10CYP2A6
SCHEMBL30469264 0.69 PDPK1 (0.60) PDPK1LOXL2ALDH1A1TSHRHSD17B10
SCHEMBL2715410 0.69 CYP2A6 (0.53) PDPK1LOXL2ALDH1A1TSHRNOS1
SCHEMBL2315490 0.69 PDPK1 (0.60) PDPK1LOXL2ALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102365277-B JUN N-terminal kinase inhibitors ELAN PHARMACEUTICALS, INC. (US) 2015-11-25 CN disclosed