SCHEMBL28825473

SCHEMBL28825473

Fc1cc(F)cc(-c2ncc(Cn3cccn3)cc2F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
KLKB1 P03952 2/20 0.36
PRKACA P17612 1/20 0.36
PRKACG P22612 1/20 0.36
PRKACB P22694 1/20 0.36
GRIN2B Q13224 2/20 0.35
KAT7 O95251 2/20 0.35
KAT6A Q92794 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KCNH2 Q12809 1/20 0.34
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825448 0.84 GAA (0.47) GAAMAPTHTTCA12CA1
SCHEMBL28825562 0.83 GAA (0.52) GAAMAPTHTTCA12CA1
SCHEMBL28825510 0.82 GRIN2B (0.52) GAAMAPTKLKB1GRIN2BKCNH2
SCHEMBL28825588 0.81 GAA (0.50) GAAMAPTHTTCA12CA1
SCHEMBL28931688 0.80 KCNH2 (0.45) GAAMAPTGRIN2BKCNH2GRIN1
SCHEMBL28825458 0.80 GAA (0.48) GAAMAPTHTTCA12CA1
SCHEMBL28949576 0.80 KCNH2 (0.49) GRIN2BKCNH2GRIN1
SCHEMBL28949592 0.78 KCNH2 (0.43) GAAMAPTHTTPRKACAPRKACG
SCHEMBL30046359 0.77 HTT (0.47) GAAMAPTHTTCA12CA1
SCHEMBL28825487 0.76 GRIN2B (0.51) GAAMAPTKLKB1GRIN2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed