SCHEMBL28825458

SCHEMBL28825458

Fc1ccccc1-c1ncc(Cn2cccn2)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
CYP11B1 P15538 3/20 0.41
CYP11B2 P19099 3/20 0.41
HTT P42858 1/20 0.39
KLKB1 P03952 2/20 0.38
GRIN2B Q13224 2/20 0.37
GRIN1 Q05586 1/20 0.37
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
KMT2A Q03164 1/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825547 0.83 GAA (0.44) GAAMAPTKLKB1GRIN2BGRIN1
SCHEMBL28825448 0.81 GAA (0.47) GAAMAPTCYP11B1CYP11B2HTT
SCHEMBL28825473 0.80 GAA (0.46) GAAMAPTHTTKLKB1GRIN2B
SCHEMBL28825562 0.80 GAA (0.52) GAAMAPTHTTKLKB1GRIN2B
SCHEMBL28825510 0.79 GRIN2B (0.52) GAAMAPTKLKB1GRIN2BGRIN1
SCHEMBL28825588 0.78 GAA (0.50) GAAMAPTHTTKLKB1GRIN2B
SCHEMBL28931688 0.77 KCNH2 (0.45) GAAMAPTGRIN2BGRIN1
SCHEMBL28949597 0.76 GAA (0.42) GAAMAPTKLKB1GRIN2BGRIN1
SCHEMBL28825653 0.75 GAA (0.44) GAAMAPTCYP11B1CYP11B2HTT
SCHEMBL28825487 0.75 GRIN2B (0.51) GAAMAPTKLKB1GRIN2BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed