SCHEMBL28825538

SCHEMBL28825538

Fc1cncc(Cn2ccc(-c3ccc(OC(F)F)c(Cl)c3)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 16/20 0.48
GRIN1 Q05586 12/20 0.48
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KCNH2 Q12809 4/20 0.39
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825518 0.91 GRIN2B (0.48) GRIN2BGRIN1KCNH2KDM4ETDP1
SCHEMBL28949575 0.89 GRIN2B (0.47) GRIN2BGRIN1MAPTSMN1; SMN2KCNH2
SCHEMBL28825478 0.89 GRIN2B (0.49) GRIN2BGRIN1KCNH2KDM4ETDP1
SCHEMBL28825482 0.87 GRIN2B (0.51) GRIN2BGRIN1KCNH2KDM4ETDP1
SCHEMBL28825441 0.84 GRIN2B (0.46) GRIN2BGRIN1MAPTSMN1; SMN2KCNH2
SCHEMBL28825585 0.81 KDM4E (0.46) GRIN2BGRIN1MAPTSMN1; SMN2KCNH2
SCHEMBL28825489 0.79 GRIN2B (0.48) GRIN2BGRIN1KCNH2
SCHEMBL28949594 0.78 MAPT (0.44) GRIN2BGRIN1MAPTSMN1; SMN2KCNH2
SCHEMBL28825447 0.77 GRIN2B (0.50) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL28931687 0.77 GRIN2B (0.48) GRIN2BGRIN1MAPTSMN1; SMN2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed