SCHEMBL28825441

SCHEMBL28825441

Fc1cncc(Cn2ccc(-c3ccc(OC(F)F)cc3)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 14/20 0.46
GRIN1 Q05586 13/20 0.46
MAPT P10636 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 2/20 0.40
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
HPGD P15428 2/20 0.40
RAB9A P51151 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNA1H O95180 1/20 0.37
CACNA1I Q9P0X4 1/20 0.37
LTA4H P09960 1/20 0.36
KCNH2 Q12809 1/20 0.36
NFKB1 P19838 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949575 0.85 GRIN2B (0.47) GRIN2BGRIN1MAPTSMN1; SMN2KCNH2
SCHEMBL28825538 0.84 GRIN2B (0.48) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL27068818 0.81 GRIN1 (0.47) GRIN2BGRIN1MAPTSMN1; SMN2
SCHEMBL28825447 0.79 GRIN2B (0.50) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL28931687 0.79 GRIN2B (0.48) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL28949591 0.78 ALDH1A1 (0.44) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL28825456 0.77 MAPT (0.56) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL28825507 0.76 SMN1; SMN2 (0.45) GRIN2BGRIN1MAPTSMN1; SMN2NPC1
SCHEMBL28825585 0.76 KDM4E (0.46) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E
SCHEMBL28825544 0.76 MAPT (0.41) GRIN2BGRIN1MAPTSMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed