SCHEMBL28825552

SCHEMBL28825552

COc1cncc(Cn2ccc(-c3ccc(C(F)(F)F)c(F)c3)n2)c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 7/20 0.58
CYP11B1 P15538 5/20 0.58
GRIN2B Q13224 10/20 0.48
GRIN1 Q05586 9/20 0.48
KDM1A O60341 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
GPR55 Q9Y2T6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949601 0.93 GRIN2B (0.49) CYP11B2CYP11B1GRIN2BGRIN1KDM1A
SCHEMBL28949561 0.88 GRIN2B (0.54) CYP11B2CYP11B1GRIN2BGRIN1KDM1A
SCHEMBL28825508 0.85 GRIN2B (0.47) CYP11B2CYP11B1GRIN2BGRIN1KDM1A
SCHEMBL28694730 0.83 GRIN2B (0.52) CYP11B2CYP11B1GRIN2BGRIN1KDM1A
SCHEMBL28825488 0.82 GRIN2B (0.50) GRIN2BGRIN1KDM1AHDAC1HDAC2
SCHEMBL28964548 0.81 SMN1; SMN2 (0.47) CYP11B2CYP11B1GRIN2BGRIN1GPR55
SCHEMBL28825494 0.80 GRIN2B (0.46) CYP11B2CYP11B1GRIN2BGRIN1
SCHEMBL28825556 0.79 GRIN2B (0.54) CYP11B2CYP11B1GRIN2BGRIN1KDM1A
SCHEMBL28825495 0.79 GRIN1 (0.47) CYP11B2CYP11B1GRIN2BGRIN1KDM1A
SCHEMBL28825464 0.76 GRIN2B (0.50) CYP11B2CYP11B1GRIN2BGRIN1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed