SCHEMBL28825653

SCHEMBL28825653

Cc1cc(Cn2cccn2)cnc1-c1ccc(F)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
GRIN2B Q13224 6/20 0.43
KLKB1 P03952 2/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
GRIN1 Q05586 4/20 0.38
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
WNT3A P56704 2/20 0.37
HDAC1 Q13547 2/20 0.37
PDE4B Q07343 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825487 0.93 GRIN2B (0.51) GAAMAPTGRIN2BKLKB1GRIN1
SCHEMBL28825448 0.91 GAA (0.47) GAAMAPTGRIN2BKLKB1CYP11B1
SCHEMBL28825554 0.89 KCNH2 (0.45) GAAMAPTGRIN2BGRIN1
SCHEMBL28825499 0.87 KCNH2 (0.47) GAAMAPTGRIN2BKLKB1GRIN1
SCHEMBL28825510 0.87 GRIN2B (0.52) GAAMAPTGRIN2BKLKB1GRIN1
SCHEMBL28949563 0.85 PDE4B (0.46) GAAMAPTGRIN2BGRIN1PDE4B
SCHEMBL28825492 0.85 KCNH2 (0.48) GRIN2BGRIN1PDE4B
SCHEMBL28949597 0.81 GAA (0.42) GAAMAPTGRIN2BKLKB1GRIN1
SCHEMBL28825588 0.81 GAA (0.50) GAAMAPTGRIN2BKLKB1CA12
SCHEMBL28825562 0.81 GAA (0.52) GAAMAPTGRIN2BKLKB1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed