SCHEMBL28825499

SCHEMBL28825499

Cc1cc(Cn2cccn2)cnc1-c1ccc(F)c(C(C)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.47
GRIN2B Q13224 14/20 0.43
GRIN1 Q05586 11/20 0.43
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
KLKB1 P03952 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825498 0.94 KCNH2 (0.48) KCNH2GRIN2BGRIN1GAAMAPT
SCHEMBL28949603 0.87 KCNH2 (0.45) KCNH2GRIN2BGRIN1
SCHEMBL28825487 0.87 GRIN2B (0.51) KCNH2GRIN2BGRIN1GAAMAPT
SCHEMBL28825653 0.87 GAA (0.44) GRIN2BGRIN1GAAMAPTKLKB1
SCHEMBL28825554 0.83 KCNH2 (0.45) KCNH2GRIN2BGRIN1GAAMAPT
SCHEMBL28825634 0.83 KCNH2 (0.43) KCNH2GRIN2BGRIN1GAAMAPT
SCHEMBL28825510 0.81 GRIN2B (0.52) KCNH2GRIN2BGRIN1GAAMAPT
SCHEMBL28825550 0.80 GAA (0.45) KCNH2GRIN2BGRIN1GAAMAPT
SCHEMBL28825555 0.80 GRIN1 (0.43) GRIN2BGRIN1GAAMAPT
SCHEMBL28825448 0.79 GAA (0.47) GRIN2BGRIN1GAAMAPTKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN claimed
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed