SCHEMBL28825843

SCHEMBL28825843

CCCCP(CCCC)c1ccccc1N(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.36
TLR8 Q9NR97 1/20 0.36
MAPT P10636 3/20 0.33
GAA P10253 2/20 0.33
ALDH1A1 P00352 2/20 0.33
TP53 P04637 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KCNH2 Q12809 2/20 0.32
CHEK1 O14757 1/20 0.32
NEK2 P51955 1/20 0.32
LIMK1 P53667 1/20 0.32
DYRK1A Q13627 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
KDM4E B2RXH2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
INSR P06213 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7930351 0.86 ALDH1A1 (0.33) HTR6TLR8MAPTGAAALDH1A1
SCHEMBL15660148 0.82 KCNH2 (0.35) TSHRSMN1; SMN2KCNH2SIGMAR1CYP1A2
SCHEMBL17529753 0.78 CA1 (0.43) TLR8ALDH1A1TP53TSHRSMN1; SMN2
SCHEMBL2848684 0.77
SCHEMBL15658031 0.76 BCHE (0.36) MAPTGAAALDH1A1TSHRSMN1; SMN2
SCHEMBL2879314 0.76 KCNH2 (0.39) ALDH1A1TP53TSHRKCNH2SIGMAR1
SCHEMBL11196033 0.76 MAPT (0.34) HTR6TLR8MAPTGAAALDH1A1
SCHEMBL11196031 0.76 MAPT (0.34) HTR6TLR8MAPTGAAALDH1A1
SCHEMBL1726391 0.75 TSHR (0.36) TLR8MAPTALDH1A1TP53TSHR
SCHEMBL5443955 0.74 CYP1A2 (0.38) MAPTTP53TSHRCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109819649-A (1S, 4S) -4- (2- (((3S, 4R) -3- fluorine tetrahydro -2H- pyrans -4- base) amino) -8- ((2,4,6- trichlorophenyl) amino) -9H- purine -9- base) and -1- hexahydrotoluene -1- formamide solid form and its application method 西格诺药品有限公司 2019-05-28 CN disclosed
CN-105324381-A Pharmaceutical formulations, procedures, solid forms and methods of use relating to 1-ethyl-7- (2-methyl-6- (1H-1,2, 4-triazol-3-yl) pyridin-3-yl) -3, 4-dihydropyrazino [2,3-b ] pyrazin-2 (1H) -one SIGNAL PHARM LLC 2016-02-10 CN disclosed