SCHEMBL28825919

SCHEMBL28825919

c1ccc(-c2nc(-c3ccc4c(c3)OCO4)c(-c3ccccn3)[nH]2)cc1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 12/20 0.82
ACVR1B P36896 3/20 0.82
MAPK14 Q16539 5/20 0.80
MAPK13 O15264 2/20 0.80
MAPK12 P53778 2/20 0.80
MAPK11 Q15759 2/20 0.80
MAPT P10636 4/20 0.77
KDM4E B2RXH2 3/20 0.77
ALDH1A1 P00352 3/20 0.77
HPGD P15428 3/20 0.77
TDP1 Q9NUW8 3/20 0.77
CSNK1A1 P48729 2/20 0.77
CSNK1D P48730 2/20 0.77
CSNK1E P49674 2/20 0.77
RIPK2 O43353 2/20 0.77
PRKD3 O94806 1/20 0.77
CYP1A2 P05177 1/20 0.77
CYP3A4 P08684 1/20 0.77
CYP2D6 P10635 1/20 0.77
MAPK1 P28482 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5139175 0.92 TGFBR1 (0.79) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL7590309 0.91 TGFBR1 (0.78) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL373558 0.91 TGFBR1 (1.00) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL4075751 0.89 TGFBR1 (0.69) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL373802 0.89 TGFBR1 (1.00) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL373248 0.89 TGFBR1 (1.00) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL4153862 0.89 TGFBR1 (0.85) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL23352241 0.88 TGFBR1 (0.73) TGFBR1ACVR1BMAPK14MAPK13MAPK12
SCHEMBL2617116 0.88 TGFBR1 (0.84) TGFBR1ACVR1BMAPK14MAPK13MAPK12
Sb-431542 SCHEMBL310028 0.88 TGFBR1 (1.00) TGFBR1ACVR1BMAPK14MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658788-A Method for preparing dopaminergic neurons 武田药品工业株式会社 2016-06-08 CN disclosed