SCHEMBL28828294

SCHEMBL28828294

COc1ccc(C2=NOC(N3CCCC3=O)C2)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.54
CYP1A2 P05177 3/20 0.49
CYP2D6 P10635 3/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C19 P33261 2/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
MIF P14174 5/20 0.49
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.45
CYP2C9 P11712 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31103576 0.84 CHRM1 (0.54) CHRM1MIF
SCHEMBL28062125 0.84 CHRM1 (0.54) CHRM1ALDH1A1NPC1RAB9ALMNA
SCHEMBL6783767 0.76 CHRM1 (0.51) CHRM1CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL28062102 0.72 CHRM1 (0.52) CHRM1CYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL13170185 0.71 CHRM1 (0.53) CHRM1
SCHEMBL6779518 0.70 CHRM1 (1.00) CHRM1
SCHEMBL19873011 0.70 MIF (0.57) CYP1A2CYP2D6CYP3A4CYP2C19MIF
SCHEMBL12294023 0.67 MIF (0.70) MIFNPC1RAB9A
SCHEMBL3981656 0.67 CYP1A2 (0.68) CYP1A2CYP2D6CYP3A4CYP2C19ALDH1A1
SCHEMBL21066132 0.66 POLB (0.56) CYP1A2CYP2D6CYP3A4CYP2C19MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105498735-A Preparation of p-tolyl/4-chlorophenyl isocyanate-modified cationic cyclodextrin chiral resolution material through click chemistry and application of chiral resolution material UNIV TIANJIN 2016-04-20 CN disclosed