SCHEMBL28830241

SCHEMBL28830241

COc1ccc(-c2n[nH]c(-c3ccc(OC)c(OC)c3)n2)cc1N

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.69
HSD17B10 Q99714 1/20 0.69
ALDH1A1 P00352 3/20 0.52
S1PR1 P21453 1/20 0.49
LCK P06239 1/20 0.48
BTK Q06187 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
NR1H2 P55055 1/20 0.48
NR1H3 Q13133 1/20 0.48
POLB P06746 1/20 0.48
TSHR P16473 1/20 0.48
GAA P10253 1/20 0.48
MPI P34949 1/20 0.48
GFER P55789 1/20 0.48
APOBEC3G Q9HC16 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28075492 0.91 KDM4E (0.62) KDM4EHSD17B10ALDH1A1S1PR1POLB
SCHEMBL28075511 0.89 KDM4E (0.58) KDM4EHSD17B10ALDH1A1S1PR1LCK
SCHEMBL28075505 0.87 NR1H2 (0.68) KDM4EHSD17B10LCKBTKADORA2A
SCHEMBL28075558 0.84 DCUN1D1 (0.51) KDM4EHSD17B10ALDH1A1LCKBTK
SCHEMBL15117081 0.84 NR1H2 (0.63) KDM4EHSD17B10ALDH1A1S1PR1ADORA2A
SCHEMBL31659621 0.83 KDM4E (0.61) KDM4EHSD17B10ALDH1A1S1PR1ADORA2A
SCHEMBL26467084 0.83 KDM4E (0.61) KDM4EHSD17B10ALDH1A1S1PR1ADORA2A
SCHEMBL28075584 0.83 KDM4E (0.48) KDM4EHSD17B10ALDH1A1LCKBTK
SCHEMBL19356089 0.80 KDM4E (0.60) KDM4EHSD17B10ALDH1A1GAAMPI
SCHEMBL26467080 0.80 ADORA2A (0.60) KDM4EHSD17B10ALDH1A1S1PR1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008557-B 3,6- diaryl-[1,2,4] triazole simultaneously purposes of [3,4-b] [1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2019-03-01 CN claimed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN claimed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106008557-A Application of 3,6-diaryl-[1,2,4] triazolo[3,4-b][1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2016-10-12 CN claimed
CN-106008557-B 3,6- diaryl-[1,2,4] triazole simultaneously purposes of [3,4-b] [1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed
CN-106008557-A Application of 3,6-diaryl-[1,2,4] triazolo[3,4-b][1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2016-10-12 CN disclosed