SCHEMBL28075558

SCHEMBL28075558

COc1ccc(-c2n[nH]c(-c3ccc4c(c3)OCO4)n2)cc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCUN1D1 Q96GG9 1/20 0.51
KDM4E B2RXH2 5/20 0.50
HSD17B10 Q99714 3/20 0.50
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ADORA2A P29274 2/20 0.44
ADORA1 P30542 1/20 0.44
MAPT P10636 4/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
KDR P35968 1/20 0.43
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28095676 0.86 DCUN1D1 (0.51) DCUN1D1KDM4EHSD17B10NPC1RAB9A
SCHEMBL28095608 0.86 DCUN1D1 (0.51) DCUN1D1KDM4EHSD17B10NPC1RAB9A
SCHEMBL28830241 0.84 KDM4E (0.69) KDM4EHSD17B10ALDH1A1ADORA2AADORA1
SCHEMBL28075557 0.82 GRK6 (0.52) DCUN1D1NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL28096083 0.79 MAPT (0.49) DCUN1D1KDM4EHSD17B10SMN1; SMN2ALDH1A1
SCHEMBL28075511 0.79 KDM4E (0.58) KDM4EHSD17B10NPC1RAB9ASMN1; SMN2
SCHEMBL17280056 0.79 DCUN1D1 (0.62) DCUN1D1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL28075492 0.78 KDM4E (0.62) KDM4EHSD17B10ALDH1A1TSHR
SCHEMBL28075505 0.78 NR1H2 (0.68) DCUN1D1KDM4EHSD17B10ADORA2AADORA1
SCHEMBL28075584 0.74 KDM4E (0.48) KDM4EHSD17B10ALDH1A1ADORA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008557-B 3,6- diaryl-[1,2,4] triazole simultaneously purposes of [3,4-b] [1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2019-03-01 CN claimed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN claimed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106008557-A Application of 3,6-diaryl-[1,2,4] triazolo[3,4-b][1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2016-10-12 CN claimed
CN-106008557-B 3,6- diaryl-[1,2,4] triazole simultaneously purposes of [3,4-b] [1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed
CN-106008557-A Application of 3,6-diaryl-[1,2,4] triazolo[3,4-b][1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2016-10-12 CN disclosed