SCHEMBL28831739

SCHEMBL28831739

CC(C)(C)OC(=O)N1CC(C(=O)O)CC1(COCc1ccccc1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
STS P08842 1/20 0.39
KLK7 P49862 2/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
S1PR5 Q9H228 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
PPARA Q07869 1/20 0.36
LIPE Q05469 1/20 0.35
USP30 Q70CQ3 1/20 0.35
KLK5 Q9Y337 1/20 0.35
ABCB1 P08183 1/20 0.35
HTT P42858 1/20 0.35
S1PR1 P21453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24175977 0.87 TACR1 (0.41) TACR1STSKLK7JAK2JAK1
SCHEMBL28566941 0.83 STS (0.38) TACR1STSKLK7JAK2JAK1
SCHEMBL28588244 0.83 PRMT5 (0.37) TACR1SMN1; SMN2STSKLK7JAK2
SCHEMBL30089180 0.79 TACR1 (0.40) TACR1NPC1RAB9ASMN1; SMN2STS
SCHEMBL24175974 0.79 TACR1 (0.40) TACR1NPC1RAB9ASMN1; SMN2STS
SCHEMBL24998912 0.79 TACR1 (0.38) TACR1NPC1RAB9ASMN1; SMN2STS
SCHEMBL19614476 0.79 TACR1 (0.45) TACR1
SCHEMBL19614478 0.79 TACR1 (0.45) TACR1
SCHEMBL703326 0.79 TACR1 (0.45) TACR1
SCHEMBL19838986 0.78 TACR1 (0.46) TACR1STSKLK7L3MBTL1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109661398-B Spiro-lactam and di-spiro-lactam NMDA receptor modulators and uses thereof 阿普廷伊克斯股份有限公司 2022-07-05 CN disclosed