Cytarabine 5'-Phosphate

Cytarabine 5'-Phosphate

SCHEMBL28833023

Nc1ccn([C@@H]2O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]2O)c(=O)n1.O=C(O)C(O)C(O)C(O)C(O)C(=O)O

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC18A2SLC6A2SLC6A3

The experimentally established mechanism targets of Cytarabine 5'-Phosphate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RY2 P41231 3/20 0.60
ST6GAL1 P15907 8/20 0.60
TSHR P16473 1/20 0.58
GLA P06280 1/20 0.58
LMNA P02545 1/20 0.58
THRB P10828 1/20 0.58
MTOR P42345 1/20 0.58
MDM2 Q00987 1/20 0.58
NCOA1 Q15788 1/20 0.58
NCOA3 Q9Y6Q9 1/20 0.58
P2RY6 Q15077 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cytarabine 5'-Phosphate SCHEMBL17934719 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL14669262 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL207204 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL18785109 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL2681941 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL16189 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL6115643 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL11217191 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL284602 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA
Cytarabine 5'-Phosphate SCHEMBL20277485 0.91 P2RY2 (0.69) P2RY2ST6GAL1TSHRGLALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507538-B Compositions and methods for cancer immunotherapy 艾杜罗生物科技公司 2018-04-06 CN disclosed
CN-106358440-A Factor vii conjugates 诺和诺德保健股份有限公司 2017-01-25 CN disclosed
CN-106029106-A Coagulation factor IX conjugates 诺和诺德保健股份有限公司 2016-10-12 CN disclosed
CN-105979972-A Factor viii conjugates 诺和诺德股份有限公司 2016-09-28 CN disclosed