SCHEMBL28833412

SCHEMBL28833412

O=c1c(CO)c(-c2ccccc2)[nH]c2ccc(Cl)cc12

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.71
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
RXFP1 Q9HBX9 1/20 0.56
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
HPGD P15428 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
ROCK2 O75116 1/20 0.51
MAP4K4 O95819 1/20 0.51
LCK P06239 1/20 0.51
CSF1R P07333 1/20 0.51
PIM1 P11309 1/20 0.51
RPS6KB1 P23443 1/20 0.51
CDK2 P24941 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28094612 0.86 PDE10A (0.71) PDE10AMEN1KMT2ARXFP1CA1
SCHEMBL13550372 0.82 KDM4E (0.62) PDE10AMEN1KMT2ARXFP1CA1
SCHEMBL6300664 0.81 PDE10A (0.60) PDE10AMEN1KMT2ARXFP1CA1
SCHEMBL28906438 0.80 TUBB4A (0.67) PDE10AMEN1KMT2ARXFP1CA1
SCHEMBL8020349 0.79 PDE10A (0.64) PDE10AMEN1KMT2ARXFP1CA1
SCHEMBL6922317 0.77 PPARG (0.66) PDE10AKDM4EALDH1A1TUBB4ATUBB
SCHEMBL29432610 0.77 DYRK1A (0.55) PDE10AMEN1KMT2AHPGDKDM4E
SCHEMBL19846959 0.77 DYRK1A (0.55) PDE10AMEN1KMT2AHPGDKDM4E
SCHEMBL16814486 0.75 KDM4E (0.57) MEN1KMT2ARXFP1CA1CA2
SCHEMBL7234310 0.75 PPARG (0.60) PDE10AHPGDCYP1A2CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008479-A Substituted pyrimidine compound serving as phosphatidylinositol 3-kinase delta inhibitor and application thereof 南京圣和药业股份有限公司 2016-10-12 CN disclosed
CN-105936635-A Compound as phosphatidylinositol 3-kinase delta inhibitor and application thereof 南京圣和药业股份有限公司 2016-09-14 CN disclosed