SCHEMBL28835192

SCHEMBL28835192

BrC1CCC2CC12.COc1ccc2ccc(=O)[nH]c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
CYP1A2 P05177 3/20 0.39
CYP2E1 P05181 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C8 P10632 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2B6 P20813 2/20 0.39
CYP2C19 P33261 2/20 0.39
CA2 P00918 1/20 0.39
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 2/20 0.39
DRD2 P14416 9/20 0.38
RXFP1 Q9HBX9 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL705545 0.81 KDM4E (0.59) KDM4ECA2MEN1POLBMAPK1
Hydrochloric Acid SCHEMBL3859534 0.79 KDM4E (0.57) KDM4ECA2MEN1POLBMAPK1
SCHEMBL878695 0.70 CA12 (0.59) KDM4ECA2MEN1POLBKMT2A
SCHEMBL18850187 0.69 ACHE (0.46) KDM4ECA2MEN1POLBMAPK1
SCHEMBL25903858 0.65 KDM4E (0.58) KDM4EMEN1POLBKMT2AALDH1A1
SCHEMBL25903978 0.65 KDM4E (0.55) KDM4ECA2MEN1POLBKMT2A
SCHEMBL24338757 0.65 CA12 (0.48) KDM4ECA2MAPK1DRD2ACHE
SCHEMBL18892613 0.65 CA12 (0.48) KDM4EMAPK1DRD2ACHEMAOB
SCHEMBL18508007 0.65 CA12 (0.48) KDM4ECYP1A2CYP3A4CYP2C19MEN1
SCHEMBL13532787 0.65 PDE3B (0.48) KDM4EMAPK1KMT2AALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061966-A Bicyclic heterocyclic derivatives as bromodomain inhibitors 奥赖恩公司 2016-10-26 CN disclosed