SCHEMBL28840490

SCHEMBL28840490

CC1=Nc2ccc(-c3ccc(C(=O)N4CCCC4)cc3)cc2C=C(C(=O)O)C1C.CCCCCN

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.45
HPGD P15428 6/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPK1 P28482 1/20 0.37
TLR7 Q9NYK1 1/20 0.36
HRH3 Q9Y5N1 5/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GBA1 P04062 1/20 0.35
TSHR P16473 1/20 0.34
PKM P14618 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
HTR1A P08908 1/20 0.33
SLC6A4 P31645 1/20 0.33
HRH1 P35367 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28145411 0.90 HPGD (0.45) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL28129050 0.84 TLR8 (0.43) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL28810372 0.82 TLR8 (0.45) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL18297270 0.78 TLR8 (0.47) TLR8HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL28145441 0.76 TLR8 (0.43) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL10325045 0.76 TLR8 (0.45) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL19119595 0.75 TLR8 (0.45) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL3021829 0.72 TLR8 (0.56) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL10325171 0.70 TLR8 (0.60) TLR8HPGDALDH1A1MEN1KMT2A
SCHEMBL27950485 0.69 TLR8 (0.46) TLR8HPGDALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103562186-B Substituted benzazepines as modulators of TOLL-like receptors 帆德制药股份有限公司 2017-02-15 CN disclosed