SCHEMBL28840671

SCHEMBL28840671

Cc1ccc2c(ccn2COCC[Si](C)(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.48
HTR2A P28223 2/20 0.48
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
DGAT1 O75907 3/20 0.39
MAPT P10636 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PRMT5 O14744 1/20 0.36
ROCK1 Q13464 1/20 0.35
NPC1 O15118 1/20 0.35
PDE10A Q9Y233 4/20 0.34
EGFR P00533 1/20 0.33
IGF1R P08069 1/20 0.33
SRC P12931 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
FLT3 P36888 1/20 0.33
EPHB4 P54760 1/20 0.33
TEK Q02763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29925168 1.00 HTR2C (0.48) HTR2CHTR2ACDK4CCND1DGAT1
SCHEMBL26728337 0.89 HTR2A (0.48) HTR2CHTR2ADGAT1PRMT5PDE10A
SCHEMBL28840665 0.84 HTR2C (0.49) HTR2CHTR2ACDK4CCND1DGAT1
SCHEMBL29924680 0.84 DGAT1 (0.36) HTR2CHTR2ADGAT1NPC1PDE10A
SCHEMBL28841058 0.84 HTR2C (0.51) HTR2CHTR2AMAPTPRMT5ROCK1
SCHEMBL28840999 0.84 DGAT1 (0.36) HTR2CHTR2ADGAT1NPC1PDE10A
SCHEMBL4493915 0.84 HTR2C (0.49) HTR2CHTR2ACDK4CCND1DGAT1
SCHEMBL29924561 0.84 HTR2C (0.51) HTR2CHTR2AMAPTPRMT5ROCK1
SCHEMBL1467091 0.84 HTR2A (0.49) HTR2CHTR2ADGAT1PRMT5ROCK1
SCHEMBL29924782 0.84 HTR2C (0.49) HTR2CHTR2ACDK4CCND1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115028655-B 2-trifluoromethyl-3-iodo-indole compound and preparation method thereof 上海大学 2024-01-16 CN claimed
CN-115028655-A 2-trifluoromethyl-3-iodine-indole compound and preparation method thereof 上海大学 2022-09-09 CN claimed
CN-115028655-B 2-trifluoromethyl-3-iodo-indole compound and preparation method thereof 上海大学 2024-01-16 CN disclosed
CN-115028655-A 2-trifluoromethyl-3-iodine-indole compound and preparation method thereof 上海大学 2022-09-09 CN disclosed