SCHEMBL28844277

SCHEMBL28844277

Cn1ncc(C(=O)N2CCOCC2)c1NC=O

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
ALDH1A1 P00352 2/20 0.46
PDE10A Q9Y233 8/20 0.45
HSD17B10 Q99714 1/20 0.45
POLB P06746 1/20 0.43
HTT P42858 1/20 0.42
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
SPR P35270 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1458472 0.75 HTT (0.52) ALDH1A1PDE10AHTT
SCHEMBL16211920 0.74 PDE10A (0.50) ALDH1A1PDE10AHTTSPR
SCHEMBL11890121 0.74 PDE10A (0.51) PDE10AHTT
SCHEMBL15767454 0.72 GAA (0.43) ALDH1A1PDE10AHSD17B10HTTSPR
SCHEMBL9926277 0.71 PDE10A (0.49) ALDH1A1PDE10AHTT
SCHEMBL4594288 0.69 CYP3A4 (0.46) CYP3A4ALDH1A1HTT
SCHEMBL7514360 0.68 SMN1; SMN2 (0.50) ALDH1A1PDE10AATML3MBTL1
SCHEMBL14368301 0.66 EPHX2 (0.59) ALDH1A1POLBHTTL3MBTL1
SCHEMBL9104445 0.65 SMN1; SMN2 (0.53) ALDH1A1PDE10APOLBHTTL3MBTL1
SCHEMBL27228782 0.65 KDM4E (0.62) ALDH1A1HTTATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164126-B The Pd catalytic couplings of pyrazole amide 豪夫迈·罗氏有限公司 2017-05-31 CN disclosed