SCHEMBL9926277

SCHEMBL9926277

Cn1ncc(C(=O)N2CCOCC2)c1C(=O)CI

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 11/20 0.49
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 2/20 0.42
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1458472 0.83 HTT (0.52) PDE10ASMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL16211920 0.82 PDE10A (0.50) PDE10ASMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL11890121 0.79 PDE10A (0.51) PDE10AHTT
SCHEMBL9926248 0.75 KDM4E (0.38) PDE10ASMN1; SMN2KDM4EALDH1A1KMT2A
SCHEMBL7514360 0.73 SMN1; SMN2 (0.50) PDE10ASMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL15767454 0.72 GAA (0.43) PDE10ASMN1; SMN2ALDH1A1HTTKMT2A
SCHEMBL9926264 0.72 PDE10A (0.39) PDE10AALDH1A1MAPT
SCHEMBL28844277 0.71 CYP3A4 (0.47) PDE10AALDH1A1HTT
SCHEMBL1458202 0.70 PDE10A (0.50) PDE10A
SCHEMBL9106126 0.70 POLB (0.49) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076430-A1 TRIAZOLOPYRIDINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2012-06-14 WO disclosed