SCHEMBL28844690

SCHEMBL28844690

NC(=O)Oc1ccc(Oc2ccc([N+](=O)[O-])cc2Cl)cc1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.71
KMT2A Q03164 8/20 0.64
MEN1 O00255 7/20 0.64
GAA P10253 1/20 0.64
PKM P14618 1/20 0.64
ALDH1A1 P00352 9/20 0.63
MAPT P10636 6/20 0.63
KDM4E B2RXH2 1/20 0.53
HGFAC Q04756 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.50
LMNA P02545 3/20 0.50
GPR55 Q9Y2T6 1/20 0.50
HSPB1 P04792 1/20 0.47
HSP90AA1 P07900 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28844657 0.88 KMT2A (0.63) PDE7AKMT2AMEN1GAAPKM
SCHEMBL29130743 0.86 HGFAC (0.62) PDE7AKMT2AMEN1GAAPKM
SCHEMBL9367473 0.83 PDE7A (0.74) PDE7AKMT2AMEN1GAAPKM
SCHEMBL11760667 0.83 PDE7A (1.00) PDE7AKMT2AMEN1GAAPKM
SCHEMBL2967458 0.83 PDE7A (0.78) PDE7AKMT2AMEN1GAAPKM
SCHEMBL3509441 0.82 PDE7A (0.68) PDE7AKMT2AMEN1GAAPKM
SCHEMBL29251429 0.82 PDE7A (0.54) PDE7AKMT2AMEN1GAAPKM
SCHEMBL11198374 0.81 PDE7A (0.76) PDE7AKMT2AMEN1GAAPKM
SCHEMBL22069562 0.80 PDE7A (0.74) PDE7AKMT2AMEN1GAAPKM
SCHEMBL4029870 0.80 PDE7A (0.73) PDE7AKMT2AMEN1GAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483366-B Indole compound and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-09-16 CN disclosed