SCHEMBL28844993

SCHEMBL28844993

OCCN1CN=C(Nc2ccc(OC(F)(F)F)cc2)c2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.41
BCR P11274 3/20 0.41
CHRNA7 P36544 1/20 0.40
P2RY1 P47900 2/20 0.39
P2RX3 P56373 1/20 0.39
MAPT P10636 5/20 0.37
MEN1 O00255 2/20 0.37
RAB9A P51151 2/20 0.37
KMT2A Q03164 2/20 0.37
EPHX2 P34913 1/20 0.37
NPC1 O15118 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GAA P10253 2/20 0.36
KDM4E B2RXH2 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
HTT P42858 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
KCNA5 P22460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19666713 0.77 ABL1 (0.39) ABL1BCRCHRNA7P2RX3MEN1
SCHEMBL20553560 0.67 ABL1 (0.45) ABL1BCRCHRNA7MAPTSMN1; SMN2
SCHEMBL11125111 0.63 CTSC (0.56) MAPTMEN1RAB9AKMT2AEPHX2
SCHEMBL1923201 0.63 MAPT (0.61) ABL1BCRCHRNA7MAPTMEN1
SCHEMBL3194551 0.63 MAPT (0.61) ABL1BCRCHRNA7MAPTMEN1
SCHEMBL20552403 0.63 DHODH (0.49) ABL1BCRMAPTDHODH
SCHEMBL1923203 0.62 MAPT (0.53) ABL1BCRP2RY1MAPTMEN1
SCHEMBL5452795 0.61 MAPT (0.51) ABL1BCRP2RX3MAPTMEN1
SCHEMBL6289309 0.61 MAPT (0.55) MAPTMEN1RAB9AKMT2AEPHX2
SCHEMBL3919027 0.61 MAPT (0.59) P2RY1MAPTEPHX2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104327084-B The small molecule myristate inhibitors and its application method of BCR ABL 达那-法伯癌症研究所 2017-06-06 CN claimed
CN-104327084-B The small molecule myristate inhibitors and its application method of BCR ABL 达那-法伯癌症研究所 2017-06-06 CN disclosed