SCHEMBL28845079

SCHEMBL28845079

O=S(=O)(c1ccc(Cn2cccn2)cc1)c1ccc(F)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
KAT7 O95251 3/20 0.40
KAT6A Q92794 3/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
GAA P10253 2/20 0.39
MAPT P10636 2/20 0.39
PIK3CA P42336 1/20 0.39
HTT P42858 1/20 0.37
NAMPT P43490 3/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
COMT P21964 3/20 0.36
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28150066 0.89 CA12 (0.49) CA12CA1CA2CA9KAT7
SCHEMBL28845062 0.82 CA12 (0.51) CA12CA1CA2CA9KAT7
SCHEMBL28149987 0.81 CA12 (0.50) CA12CA1CA2CA9KAT7
SCHEMBL28148776 0.80 CA12 (0.49) CA12CA1CA2CA9KAT7
SCHEMBL28148744 0.80 CA12 (0.49) CA12CA1CA2CA9KAT7
SCHEMBL28150075 0.80 CA12 (0.49) CA12CA1CA2CA9KAT7
SCHEMBL28149998 0.80 CA12 (0.51) CA12CA1CA2CA9KAT7
SCHEMBL28149935 0.79 CA12 (0.50) CA12CA1CA2CA9KAT7
SCHEMBL28844823 0.78 CA12 (0.58) CA12CA1CA2CA9KAT7
SCHEMBL22446082 0.76 CA12 (0.52) CA12CA1CA2CA9KAT7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103384668-B compounds and compositions for inhibition of NAMPT 福马TM有限责任公司 2017-05-31 CN claimed