SCHEMBL28845657

SCHEMBL28845657

CC(C)NC(=O)c1ccc(Nc2ccnc3cc(C(F)(F)F)ccc23)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 3/20 0.57
RIPK2 O43353 2/20 0.49
EPHB6 O15197 1/20 0.49
ABL1 P00519 1/20 0.49
LCK P06239 1/20 0.49
EPHA1 P21709 1/20 0.49
EPHA8 P29322 1/20 0.49
TXK P42681 1/20 0.49
COQ8A Q8NI60 1/20 0.49
NLK Q9UBE8 1/20 0.49
DNMT1 P26358 3/20 0.49
DNMT3A Q9Y6K1 2/20 0.49
HDAC3 O15379 1/20 0.49
ACHE P22303 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28845648 0.90 NPSR1 (0.56) GAKRIPK2EPHB6ABL1LCK
Hydrochloric Acid SCHEMBL11735917 0.87 GAK (0.56) GAKRIPK2EPHB6ABL1LCK
SCHEMBL10664310 0.85 GAK (0.57) GAKRIPK2EPHB6ABL1LCK
SCHEMBL28845677 0.85 GAK (0.54) GAKRIPK2EPHB6ABL1LCK
SCHEMBL29822705 0.84 GAK (0.56) GAKRIPK2EPHB6ABL1LCK
Hydrochloric Acid SCHEMBL11523664 0.84 GAK (0.56) GAKRIPK2EPHB6ABL1LCK
SCHEMBL11737693 0.83 GAK (0.55) GAKRIPK2EPHB6ABL1LCK
Hydrochloric Acid SCHEMBL11738528 0.83 GAK (0.55) GAKRIPK2EPHB6ABL1LCK
Hydrochloric Acid SCHEMBL10625573 0.83 GAK (0.55) GAKRIPK2EPHB6ABL1LCK
SCHEMBL28845671 0.83 GAK (0.53) GAKRIPK2EPHB6ABL1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN claimed
CN-114773267-B [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2024-01-26 CN disclosed
CN-114773267-A [ (7-trifluoromethyl quinoline-4-yl) amino ] benzamide compound and preparation and application thereof 沈阳药科大学 2022-07-22 CN disclosed