SCHEMBL28845869

SCHEMBL28845869

COC(=O)c1ccc(-c2ccc(N3CCN(C)CC3)c([N+](=O)[O-])c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.62
ALDH1A1 P00352 3/20 0.62
KDM4E B2RXH2 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
HPGD P15428 1/20 0.62
CYP2C19 P33261 1/20 0.62
WDR5 P61964 4/20 0.61
SMN1; SMN2 Q16637 5/20 0.60
LMNA P02545 2/20 0.60
MAPK1 P28482 2/20 0.58
GAA P10253 2/20 0.57
POLB P06746 1/20 0.55
SIRT6 Q8N6T7 1/20 0.55
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4289177 0.90 WDR5 (0.69) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL29891470 0.87 MAPT (0.59) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL29892052 0.86 WDR5 (0.62) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL29891273 0.84 WDR5 (0.54) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL29891093 0.84 WDR5 (0.59) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL23292304 0.83 WDR5 (0.62) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL29994410 0.83 WDR5 (0.62) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL28845856 0.81 SMN1; SMN2 (0.61) MAPTALDH1A1KDM4ECYP1A2CYP2D6
SCHEMBL29891443 0.81 KDM4E (0.62) MAPTALDH1A1KDM4EHPGDWDR5
SCHEMBL1657077 0.80 SMN1; SMN2 (0.64) MAPTALDH1A1KDM4ECYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed