SCHEMBL28846345

SCHEMBL28846345

NC(=O)c1ccc(NC[C@H]2COCCO2)c([N+](=O)[O-])c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.75
MAPT P10636 10/20 0.67
MEN1 O00255 6/20 0.67
HCAR3 P49019 1/20 0.61
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 6/20 0.54
SMN1; SMN2 Q16637 6/20 0.54
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
LMNA P02545 4/20 0.52
GAA P10253 1/20 0.52
CRHBP P24387 1/20 0.52
CRHR2 Q13324 1/20 0.52
PKM P14618 1/20 0.51
MAPK1 P28482 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
HPGD P15428 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28846346 1.00 KMT2A (0.75) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL20798382 0.90 HCAR3 (0.74) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL20798381 0.90 HCAR3 (0.74) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL19858272 0.82 HCAR3 (0.52) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL30921528 0.82 KMT2A (0.71) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL29262732 0.82 KMT2A (0.71) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL4966338 0.82 HCAR3 (0.54) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL4966333 0.82 HCAR3 (0.54) KMT2AMAPTMEN1HCAR3KDM4E
SCHEMBL1810940 0.81 MAPT (0.66) KMT2AMAPTMEN1HCAR3ALDH1A1
SCHEMBL16037933 0.81 MAPT (0.66) KMT2AMAPTMEN1HCAR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114073703-B Compositions and methods for treating nonalcoholic steatohepatitis 苏州亚盛药业有限公司 2022-12-30 CN disclosed
CN-114073703-A Compositions and methods for treating nonalcoholic steatohepatitis 苏州亚盛药业有限公司 2022-02-22 CN disclosed