SCHEMBL28847737

SCHEMBL28847737

c1ccc(-c2ccc3c(ccc4ccc(-c5ccccc5)cc43)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.53
ESR2 Q92731 5/20 0.53
ALDH1A1 P00352 1/20 0.52
HIF1A Q16665 1/20 0.52
CYP1B1 Q16678 1/20 0.52
HSD17B10 Q99714 1/20 0.52
GPR84 Q9NQS5 1/20 0.47
HSD17B1 P14061 3/20 0.47
HSD17B2 P37059 3/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2B6 P20813 1/20 0.47
CYP2C19 P33261 1/20 0.47
BACE1 P56817 1/20 0.46
PGR P06401 1/20 0.44
HPRT1 P00492 1/20 0.44
NPC1 O15118 1/20 0.44
CDK4 P11802 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30703158 0.93 ESR1 (0.58) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL2724557 0.93 ESR1 (0.58) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL1987912 0.93 ESR1 (0.58) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL2723055 0.91 ALDH1A1 (0.58) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL19558296 0.91 ESR1 (0.50) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL3005121 0.91 ESR1 (0.56) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL30960425 0.91 ESR1 (0.54) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL3695546 0.91 ESR1 (0.54) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL6559203 0.88 ALDH1A1 (0.61) ESR1ESR2ALDH1A1HIF1ACYP1B1
SCHEMBL26478504 0.87 ESR1 (0.44) ESR1ESR2ALDH1A1HIF1ACYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107250150-B Chlolic acid derivatives and preparation method thereof and medical usage 江苏豪森药业集团有限公司 2019-11-22 CN disclosed
CN-107250150-A Cholic acid derivative and preparation method and medical application thereof 江苏豪森药业集团有限公司 2017-10-13 CN disclosed