SCHEMBL28848348

SCHEMBL28848348

Cc1c(C(F)(F)F)cc(C(=O)O)c(Cl)c1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C19 P33261 2/20 0.48
TSHR P16473 3/20 0.38
NOTUM Q6P988 3/20 0.38
PKM P14618 1/20 0.38
TDP1 Q9NUW8 2/20 0.37
CYP3A4 P08684 2/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HIF1A Q16665 1/20 0.37
TXNRD1 Q16881 1/20 0.37
TXNRD3 Q86VQ6 1/20 0.37
TXNRD2 Q9NNW7 1/20 0.37
CDK2 P24941 1/20 0.37
EPAS1 Q99814 2/20 0.36
MEN1 O00255 1/20 0.36
TTR P02766 1/20 0.36
PPOX P50336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28848323 0.83 TSHR (0.38) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL450176 0.81 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL10631372 0.80 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL10628873 0.80 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL2612651 0.80 TSHR (0.53) ALDH1A1TSHRTDP1CYP3A4HPGD
SCHEMBL30855346 0.80 TSHR (0.53) ALDH1A1TSHRTDP1CYP3A4HPGD
SCHEMBL10986975 0.79 TSHR (0.53) ALDH1A1CYP1A2CYP2C19TSHRTDP1
SCHEMBL9550142 0.79 TSHR (0.45) ALDH1A1CYP1A2CYP2C19TSHRNOTUM
SCHEMBL27621308 0.77 TDP1 (0.39) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR
SCHEMBL7012924 0.75 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2D6CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114957235-B Benzothiazinone derivatives, preparation method and application thereof 四川大学华西医院 2023-10-24 CN disclosed
CN-114957235-A Benzothiazinone derivative and preparation method and application thereof 四川大学华西医院 2022-08-30 CN disclosed