SCHEMBL28848700

SCHEMBL28848700

Brc1ccnc(-n2cnc(C3CC3)c2)c1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 14/20 0.35
GRM5 P41594 3/20 0.35
GRM1 Q13255 2/20 0.32
PDE10A Q9Y233 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
NLRP3 Q96P20 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20743016 0.78 PDE10A (0.45) MAP3K5PDE10A
SCHEMBL28652012 0.77 KDM4C (0.55)
SCHEMBL28660342 0.76 KDM4C (0.43) MAP3K5PDE10A
SCHEMBL25316841 0.76 MAP3K5 (0.47) MAP3K5NPC1RAB9ANLRP3
SCHEMBL21461042 0.76 MAP3K5 (0.42) MAP3K5
SCHEMBL30352583 0.76 MAP3K5 (0.47) MAP3K5NPC1RAB9ANLRP3
SCHEMBL28392385 0.74 CYP2E1 (0.42)
SCHEMBL25316032 0.74 NPC1 (0.53) MAP3K5NPC1RAB9ANLRP3
SCHEMBL28848718 0.74 MAP3K5 (0.38) MAP3K5GRM5NPC1RAB9A
SCHEMBL25318462 0.74 MAP3K5 (0.42) MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110036005-B Amide derivatives and their use in medicine 广东东阳光药业有限公司 2022-09-27 CN disclosed